Parte II: Risultati della ricerca


Sezione D - Produzione scientifica


Sezione E - Internazionalizzazione

Contributo in rivista

Le pubblicazioni visualizzate in questo quadro sono ordinate per Classificazione, Titolo. Vengono visualizzati gli autori appartenenti al Dipartimento. Per consultare la lista completa delle informazioni relative alle pubblicazioni cliccare sul nome autori. Il campo "Provenienza del dato", se presente, indica il CRIS di Ateneo di provenienza del dato.

N.ClassificazionePubblicazione
1. Articolo in rivista

CAROCCI A (2011) "1-Pentanoyl-N-{[2’-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}- pyrrolidine-2-carboxamide: Investigation of Structural Variations"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
2. Articolo in rivista

CATALANO A (2011) "1-Pentanoyl-N-{[2’-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-pyrrolidine-2-carboxamide: Investigation of Structural Variations"

Scopus: 2-s2.0-80052414491 Web of Science: WOS:000295293800007 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
3. Articolo in rivista

FRANCHINI C (2011) "1-Pentanoyl-N-{[2’-(1H-tetrazol-5-yl)biphenyl-4-yl]methyl}-pyrrolidine-2-carboxamide: Investigation of Structural Variations"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
4. Articolo in rivista

NISO M (2011) "Analogues of sigma Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)- propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
5. Articolo in rivista

LACIVITA E (2011) "Analogues of s Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers"

Scopus: 2-s2.0-79951840503 Web of Science: WOS:000287338200011 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
6. Articolo in rivista

ABATE C (2011) "Analogues of s Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) with Added Polar Functionality and Reduced Lipophilicity for Potential Use as Positron Emission Tomography Radiotracers"

Scopus: 2-s2.0-79951840503 Web of Science: WOS:000287338200011 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
7. Articolo in rivista

Carotti A (2011) "BCR-ABL inhibitors in chronic myeloid leukemia: process chemistry and biochemical profile"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
8. Articolo in rivista

DE CANDIA M (2011) "Biarylmethoxy isonipecotanilides as potent and selective inhibitors of blood coagulation factor Xa"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
9. Articolo in rivista

Nicolotti O (2011) "Biarylmethoxy isonipecotanilides as potent and selective inhibitors of blood coagulation factor Xa"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
10. Articolo in rivista

ALTOMARE C. (2011) "Biarylmethoxy isonipecotanilides as potent and selective inhibitors of blood coagulation factor Xa"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
11. Articolo in rivista

ANTONIO LAGHEZZA (2011) "Biphenyl Sulfonylamino Methyl Bisphosphonic Acids as Inhibitors of Matrix Metalloproteinases and Bone Resorption"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
12. Articolo in rivista

LOIODICE F (2011) "Biphenyl sulfonylamino methyl bisphosphonic acids as inhibitors of matrix metalloproteinases and bone resorption"

Scopus: 2-s2.0-79959748552 Web of Science: WOS:000292212100013 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
13. Articolo in rivista

TORTORELLA P (2011) "Biphenyl sulfonylamino methyl bisphosphonic acids as inhibitors of matrix metalloproteinases and bone resorption"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
14. Articolo in rivista

CELLAMARE S (2011) "Carbamate Prodrug Concept for Hydroxamate HDAC Inhibitors"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
15. Articolo in rivista

CAROTTI A (2011) "Carbamate prodrug concept for hydroxamate HDAC"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
16. Articolo in rivista

Nicolotti O (2011) "D184E MUTATION IN AQUAPORIN-4 GENE IMPAIRS WATER PERMEABILITY AND LINKS TO DEAFNESS"

Web of Science: WOS:000297140700009 Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
17. Articolo in rivista

Carotti A (2011) "D184E mutation in aquaporin-4 gene impairs water permeability and links to deafness"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
18. Articolo in rivista

CORBO F (2011) "DESIGN AND SYNTHESIS OF THIENYLPYRIDYL GARLANDS AS NON-PEPTIDIC ALPHA HELIXMIMETICS AND POTENTIAL PROTEIN-PROTEIN INTERACTIONS DISRUPTORS"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
19. Articolo in rivista

Capogrosso R (2011) "Daily Treatment with SMTC1100, a Novel Small Molecule Utrophin Upregulator, Dramatically Reduces the Dystrophic Symptoms in the mdx Mouse"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
20. Articolo in rivista

DE LUCA A (2011) "Daily treatment with SMTC1100, a novel small molecule utrophin upregulator, dramatically reduces the dystrophic symptoms in the mdx mouse"

Scopus: 2-s2.0-79955867741 Web of Science: WOS:000290305600014 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
21. Articolo in rivista

Cozzoli A (2011) "Daily treatment with SMTC1100, a novel small molecule utrophin upregulator, dramatically reduces the dystrophic symptoms in the mdx mouse"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
22. Articolo in rivista

FRANCHINI C (2011) "Design and synthesis of thienylpyridyl garlands as non-peptidic alpha helix mimetics and potential protein–protein interactions disruptors"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
23. Articolo in rivista

Nicolotti O (2011) "Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Aromatase Inhibitors Selective over 17-alpha-Hydroxylase/C17-20 Lyase"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
24. Articolo in rivista

PISANI L (2011) "Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Aromatase Inhibitors Selective over 17-alpha-hydroxylase/C17-20 lyase"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
25. Articolo in rivista

CATTO M (2011) "Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Aromatase Inhibitors Selective over 17-alphahydroxylase/C17-20 lyase"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
26. Articolo in rivista

LEONETTI F (2011) "Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Aromatase Inhibitors Selective over 17-a-Hydroxylase/C17-20 Lyase"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
27. Articolo in rivista

CAROTTI A (2011) "Design, Synthesis, and Biological Evaluation of Imidazolyl Derivatives of 4,7-Disubstituted Coumarins as Selective Aromatase Inhibitors"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
28. Articolo in rivista

CAROTTI A (2011) "Design, synthesis and pharmacobiological evaluation of novel acrylic acid derivatives acting as lipoxygenase and cyclooxygenase inhibitors with antioxidant and anti-inflammatory activities"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
29. Articolo in rivista

Nicolotti O (2011) "Design, synthesis and pharmacobiological evaluation of novel acrylic acid derivatives acting as lipoxygenase and cyclooxygenase-1 inhibitors with antioxidant and anti-inflammatory activities"

Web of Science: WOS:000286905400023 Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
30. Articolo in rivista

STEFANACHI A (2011) "Design, synthesis, and biological evaluation of imidazolyl derivatives of 4,7-disubstituted coumarins as aromatase inhibitors selective over 17-alpha-hydroxylase/C17-20 lyase"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
31. Articolo in rivista

LEONETTI F (2011) "Discovery of a potent and selective hetero-bivalent AChE inhibitor via bioisosteric replacement"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
32. Articolo in rivista

ABATE C (2011) "Effects of PB190 and PB212, new sigma receptor ligands, on glucocorticoid receptor-mediated gene transcription in LMCAT cells"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
33. Articolo in rivista

BERARDI F (2011) "Effects of PB190 and PB212, new sigma receptor ligands, on glucocorticoid receptor-mediated gene transcription in LMCAT cells"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
34. Articolo in rivista

PERRONE R (2011) "Fluorescent Derivatives of s Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a Tool for Uptake and Cellular Localization Studies in Pancreatic Tumor Cells"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
35. Articolo in rivista

ABATE C (2011) "Fluorescent Derivatives of s Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a Tool for Uptake and Cellular Localization Studies in Pancreatic Tumor Cells"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
36. Articolo in rivista

NISO M (2011) "Fluorescent Derivatives of s Receptor Ligand 1-Cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a Tool for Uptake and Cellular Localizzation Studies in Pancreatic Tumor Cells"

Scopus: 2-s2.0-80051862694 Web of Science: WOS:000294077300017 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
37. Articolo in rivista

BERARDI F (2011) "Fluorescent derivatives of σ receptor ligand 1-cyclohexyl-4-[3-(5-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)propyl]piperazine (PB28) as a tool for uptake and cellular localization studies in pancreatic tumor cells"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
38. Articolo in rivista

Imbrici P (2011) "Genetic inactivation of Kcnj16 identifies Kir5.1 as an important determinant of neuronal PCO2/pH sensitivity"

Scopus: 2-s2.0-78650952629 Web of Science: WOS:000285782800021 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
39. Articolo in rivista

CAROTTI A (2011) "Homo- and Hetero-dimeric Bis-quaternary Heterocyclic Ammonium Salts as Potent Acetyl- and Butyryl-cholinesterase Inhibitors: A Systematic Investigation of the Influence of Linker and Cationic Heads Over Affinity and Selectivity"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
40. Articolo in rivista

PISANI L (2011) "Homo- and Hetero-dimeric bis-Quaternary Heterocyclic Ammonium Salts as Potent Acetyl- and Butyryl-cholinesterase Inhibitors: A Systematic Investigation of the Influence of Linker and Cationic Heads Over Affinity and Selectivity"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
41. Articolo in rivista

Nicolotti O (2011) "Homodimeric Bis-Quaternary Heterocyclic Ammonium Salts as Potent Acetyl- and Butyrylcholinesterase Inhibitors: A Systematic Investigation of the Influence of Linker and Cationic Heads over Affinity and Selectivity"

Web of Science: WOS:000289697800005 Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
42. Articolo in rivista

CATTO M (2011) "Homodimeric bis-Quaternary Heterocyclic Ammonium Salts as Potent Acetyl- and Butyrylcholinesterase Inhibitors: A Systematic Investigation of the Influence of Linker and Cationic Heads Over Affinity and Selectivity"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
43. Articolo in rivista

LEONETTI F (2011) "Homodimeric bis-quaternary heterocyclic ammonium salts as potent acetyl- and butyrylcholinesterase inhibitors: a systematic investigation of the influence of linker and cationic heads over affinity and selectivity"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
44. Articolo in rivista

Leopoldo M (2011) "Increase of Capsaicin-Induced Trigeminal Fos-Like Immunoreactivity by 5-HT(7) Receptors."

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
45. Articolo in rivista

Lacivita E (2011) "Increase of Capsaicin-Induced Trigeminal Fos-Like Immunoreactivity by 5-HT(7) Receptors. "

Scopus: 2-s2.0-81255124339 Web of Science: WOS:000297214800006 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
46. Articolo in rivista

Leonetti F (2011) "Insights into the complex formed by matrix metalloproteinase-2 and alloxan inhibitors: molecular dynamics simulations and free energy calculations"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
47. Articolo in rivista

Denora N (2011) "Methotrexate-Loaded Chitosan- and Glycolchitosan-Based Nanoparticles: A Promising Strategy for the Administration of the Anticancer Drug to Brain Tumors"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
48. Articolo in rivista

TRAPANI A (2011) "Methotrexate-loaded Chitosan- and Glycolchitosan-based nanoparticles: a promising strategy for the administration of the anticancer drug to brain tumors"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
49. Articolo in rivista

MANGIATORDI G (2011) "Modeling proton transfer in imidazole-like dimers: A density functional theory study"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
50. Articolo in rivista

LAQUINTANA V (2011) "New Fluorescent Probes Targeting the Mitochondrial-Located Translocator Protein 18 kDa (TSPO) as Activated Microglia Imaging Agents"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
51. Articolo in rivista

TRAPANI G (2011) "New Fluorescent Probes Targeting the Mitochondrial-Located Translocator Protein 18 kDa (TSPO) as Activated Microglia Imaging Agents"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
52. Articolo in rivista

Denora N (2011) "New Fluorescent Probes Targeting the Mitochondrial-Located Translocator Protein 18 kDa (TSPO) as Activated Microglia Imaging Agents"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
53. Articolo in rivista

TRAPANI A (2011) "New fluorescent probes targeting the mithocondrial located Translocator protein 18 KDa(TSPO) as activated microglia imaging agents"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/09
54. Articolo in rivista

DEGENNARO L (2011) "Nitrogen Dynamics and Reactivity of Chiral Aziridines: Generation of Configurationally Stable Aziridinyllithium Compounds"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/06
55. Articolo in rivista

LUISI R (2011) "Nitrogen Dynamics and Reactivity of Chiral Aziridines: Generation of Configurationally Stable Aziridinyllithiums"

Scopus: 2-s2.0-79954614820 Web of Science: WOS:000290213100009 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/06
56. Articolo in rivista

COLABUFO N (2011) "Novel Potent and Selective Sigma Ligands: Evaluation of Their Agonist and Antagonist Properties"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
57. Articolo in rivista

BERARDI F (2011) "Seroronin 5-HT7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
58. Articolo in rivista

LACIVITA E (2011) "Serotonin 5-HT7 receptor agents: Structure-activity relationships and potential therapeutic applications in central nervous system disorders"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
59. Articolo in rivista

LEOPOLDO M (2011) "Serotonin 5-HT7 receptor agents: structure-activity relationships and potential therapeutic applications in central nervous system disorders"

Scopus: 2-s2.0-79151477312 Web of Science: WOS:000287949900002 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
60. Articolo in rivista

PERRONE R (2011) "Serotonin 5-HT7 receptor agents: structure-activity relationships and potential therapeutic applications in central nervous system disorders"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
61. Articolo in rivista

LEONETTI F (2011) "Strategies of multi-objective optimization in drug discovery and development"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
62. Articolo in rivista

CAROTTI A (2011) "Targeting Monoamine Oxidases with Multipotent Ligands: An Emerging Strategy in the Search of New Drugs Against Neurodegenerative Diseases"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: CHIM/08
63. Abstract in rivista

De Luca A (2011) "Cyclic nucleotide signalling pathways as a potential druggable target for enhancing regeneration potential in dystrophic skeletal muscle"

Web of Science: WOS:000295955900239 Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
64. Abstract in rivista

Cozzoli A (2011) "Evaluation of potential efficacy of GLPG0492, a novel selective androgen receptor modulator, in the exercised-mdx mouse model: Comparison with a-methyl prednisolone and nandrolone"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
65. Abstract in rivista

De Luca A (2011) "Evaluation of potential efficacy of GLPG0492, a novel selective androgen receptor modulator, in the exercised-mdx mouse model: Comparison with a-methyl prednisolone and nandrolone"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
66. Abstract in rivista

Capogrosso R (2011) "Evaluation of potential efficacy of GLPG0492, a novel selective androgen receptor modulator, in the exercised-mdx mouse model: comparison with a-methyl prednisolone and nandrolone."

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
67. Abstract in rivista

Imbrici P (2011) "The Kir5.1 Potassium Channel is an Important Determinant of Neuronal PCO2/pH Sensitivity."

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
68. Abstract in rivista

De Luca A (2011) "Toward the identification of druggable pathways involved in disease-related fatigue in Duchenne muscular dystrophy: In vivo and ex vivo studies in dystrophic mdx mice"

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
69. Abstract in rivista

Capogrosso R (2011) "Toward the identification of druggable pathways involved in disease-related fatigue in Duchenne muscular dystrophy: in vivo and ex vivo studies in dystrophuc mdx mice."

Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14
70. Abstract in rivista

Cozzoli A (2011) "Toward the identi¿cation of drugg able pathways involved in disease-related fatigue in Duchenne muscular dystrophy: In vivo and ex vivo studies in dystrophic mdx mice"

Lingua: ENG Co-autori stranieri: Si SSD di afferenza degli autori del Dipartimento: BIO/14


Sezione F - Docenti senza produzione scientifica


Sezione G - Bandi competitivi


Sezione H - Responsabilità e riconoscimenti scientifici