IL PORTALE per la RICERCA dei DIPARTIMENTI

La Regina G., Silvestri R. (2011) "1-Aryl-5-(1H-pyrrol-1-yl)-1H-pyrazole-3-carboxamide: an effective scaffold for the design of either CB1 or CB2 receptor ligands."

FABRIZI G., GOGGIAMANI A. (2011) "2,5,7-Trisubstituted benzo[b]furans through a copper- and/or palladium-catalyzed assembly and functionalization process"

Marianecci C, Carafa M, Rinaldi F, Di Meo C, Matricardi P, Coviello T (2011) "A New Vesicle-loaded Hydrogel System Suitable for Topical Applications: Preparation and Characterization"

Curcio D (2011) "A SIMPLIFIED PROCEDURE FOR GC/C/IRMS ANALYSIS OF UNDERIVATIZED 19-NORANDROSTERONE IN URINE FOLLOWING HPLC PURIFICATION"

Rossella Fioravanti, Adriana Bolasco (2011) "A chromatographic study on the exceptional enantioselectivity of cellulose tris(4-methylbenzoate) towards C5-chiral 4,5-dihydro-(1H)-pyrazole derivatives"

Biava M. (2011) "A fast virtual screening approach to identify structurally diverse inhibitors of trypanothione reductase"

CRESTONI M. E, S. FORNARINI (2011) "A neutralization-reionization and reactivity mass spectrometry study of the generation of neutral hydroxymethylene"

ROTILI D., MAI A (2011) "A photoreactive small-molecule probe for 2-oxoglutarate oxygenases."

L. SCIPIONE, S. TORTORELLA, D. DE VITA (2011) "Activity of Drugs Against Dormant Mycobacterium tuberculosis"

DI MEO C, COVIELLO T, MATRICARDI P (2011) "Anisotropic enhanced water diffusion in scleroglucan gel tablets"

BARBA M, BOTTA B, CALCATERRA A (2011) "Antioxidant Properties of Aminoethylcysteine Ketimine Decarboxylated Dimer: A Review"

Mai A, Valente S (2011) "Application of 3 µm particle-based amylose-derived chiral stationary phases for the enantioseparation of potential histone deacetylase inhibitors."

Claudio Villani (2011) "Application of circular dichroism spectroscopy in the study of mixed-valence asymmetric ruthenium polypyridyl complexes "

Mazzei F. (2011) "Aptamer-based and DNAzyme-based biosensors for environmental monitoring"

F. MAZZEI (2011) "Azurin modulates the association of Mdm2 with p53: SPR evidence from interaction of the full-length proteins."

Rino Ragno (2011) "Beneficial effect of Mentha suaveolens essential oil in the treatment of vaginal candidiasis assessed by real-time monitoring of infection"

COVIELLO T, MATRICARDI P (2011) "Biodegradable IPNs based on oxidized alginate and dextran-HEMA for controlled release of proteins"

Dante Rotili, Antonello Mai (2011) "Biological Effects of MC2050, a Quinazoline-Based PARP-1 Inhibitor, in Human Neuroblastoma and EBV-Positive Burkitt's Lymphoma Cells"

Maria Elisa Crestoni (2011) "Biomimetic Oxidation Reactions of a Naked Manganese(V)–Oxo Porphyrin Complex"

GABRIELE FAVERO, F. MAZZEI (2011) "Characterization and application of a Diamine Oxidase from Lathyrus sativus as Component of an Electrochemical Biosensor for the Determination of Biogenic Amines in wine and beer"

L.Mannina (2011) "Characterization of mono-varietal oils from Molise (Gentile di Larino and Oliva nera di Colletorto) through an advanced statistical procedure applied to data acquired by sensory, conventional, gas chromatographic and nuclear magnetic resonance analysis"

FEDERICO PEPI, STEFANIA GARZOLI, PIERLUIGI GIACOMELLO, RINO RAGNO, GABRIELE FAVERO, F. MAZZEI (2011) "Chemically Modified Multiwalled Carbon Nanotubes Electrodes with Ferrocene Derivatives through Reactive Landing"

M. PIERINI (2011) "Chemoselective C-4 Aerobic Oxidation of Catechin Derivatives Catalyzed by the Trametes villosa Laccase/1-Hydroxybenzotriazole System: Synthetic and Mechanistic Aspects"

Luisa Mannina (2011) "Conversion of the Mycotoxin Patulin to the Less Toxic Desoxypatulinic Acid by the Biocontrol Yeast Rhodosporidium kratochvilovae Strain LS11 "

FABRIZI G, A. GOGGIAMANI (2011) "Copper catalysis in the construction of indole and benzo[b]furan rings"

Giuseppe La Regina, Antonio Coluccia, Romano Silvestri (2011) "Design and Synthesis of 2-Heterocyclyl-3-arylthio-1H-indoles as Potent Tubulin Polymerization and Cell Growth Inhibitors with Improved Metabolic Stability"

Nicoletta Desideri (2011) "Design, synthesis and in vitro evaluation of novel chroman-4-one, chroman, and 2H-chromene derivatives as human rhinovirus capsid-binding inhibitors"

Riccarda Antiochia (2011) "Determination of biogenic amines in wines by HPLC-UV and LC-ESI-MS: a comparative study"

COVIELLO T (2011) "Determination of the sorption efficiency of poly(vinyl alcohol)/scleroglucan cryogels, against Cu(2+) ions"

BIAVA M, POCE G, ALFONSO S (2011) "Developing Pyrrole-Derived Antimycobacterial Agents: a Rational Lead Optimization Approach."

ROTILI D, A. MAI (2011) "Diarylpyrimidine-Dihydrobenzyloxopyrimidine Hybrids: New, Wide-Spectrum Anti-HIV-1 Agents Active at (Sub)-Nanomolar Level."

Di Santo R (2011) "Diketo acids derivatives as dual inhibitors of human immunodeficiency virus type 1 integrase and the reverse transcriptase RNase H domain."

Baiocco P (2011) "Discovery of (7R)-14-Cyclohexyl-7-{[2-(dimethylamino)ethyl](methyl) amino}-7,8-dihydro-6H-indolo[1,2-e][1,5]benzoxazocine-11-carboxylic Acid (MK-3281), a Potent and Orally Bioavailable Finger-Loop Inhibitor of the Hepatitis C Virus NS5B Polymerase"

A. MAI (2011) "Discovery, Synthesis, and Pharmacological Evaluation of Spiropiperidine Hydroxamic Acid Based Derivatives as Structurally Novel Histone Deacetylase (HDAC) Inhibitors."

Enrico Morera, Giorgio Ortar (2011) "Discussion Addendum for: Palladium-Catalyzed Reduction of Vinyl Trifluoromethanesulfonates to Alkenes: Cholesta-3,5-DieneOrganic Syntheses"

S. STRANGES (2011) "Dissociative double photoionization of benzene molecules in the 26–33 eV energy range"

Stefano Stranges (2011) "Dissociative double photoionization of singly deuterated benzene molecules in the 26-33 eV energy range"

R. Silvestri, G. La Regina (2011) "Drug-induced inhibition of tubulin polymerization induces mitochondrion-mediated apoptosis in yeast."

CARRADORI S., SECCI D., MAI A. (2011) "EPIGENETIC MODULATION OF PGC-1a ACTIVITY BY GCN5 INHIBITORS: WO2010007085"

I. D'ACQUARICA, F. GASPARRINI, M. PIERINI, P. SIMONE, C. VILLANI (2011) "Efficient organic monoliths prepared by gamma-radiation induced polymerization in the evaluation of histone deacetylase inhibitors by capillary(nano)-high performance liquid chromatography and ion trap mass spectrometry."

T. COVIELLO (2011) "Encapsulation of Cwp84 into pectin beads for oral vaccination against Clostridium difficile"

M. BIAVA, POCE G (2011) "Enlarging the NSAIDs Family: Ether, Ester and Acid Derivatives of the 1,5-Diarylpyrrole Scaffold as Novel Anti-Inflammatory and Analgesic Agents"

Carlotta Marianecci (2011) "Existence of hybrid structures in cationic liposome/DNA complexes revealed by their interaction with plasma proteins"

C. Fraschetti, M. Pierini, C. Villani, F. Gasparrini, A. Filippi (2011) "Facial control of gas-phase enantioselectivity of strapped tetra-amide macrocycles"

Sergio Valente (2011) "Facile synthesis of 4-acetyl-coumarins, -thiocoumarin and -quinolin-2(1H)-one via very high a-regioselective Heck coupling on tosylates"

Carlotta Marianecci, Maria Carafa (2011) "Factors Determining the Superior Performance of Lipid/DNA/Protammine Nanoparticles over Lipoplexes"

G. Fabrizi, A. Goggiamani, A. Iazzetti (2011) "Functionalized 2,3-dihydrofurans via palladium-catalyzed oxyarylation of a-allyl-ß-ketoesters"

Biava M. (2011) "Fyn kinase in brain diseases and cancer: the search for inhibitors."

Antonello Mai (2011) "Gold drug auranofin restricts the viral reservoir in the monkey AIDS model and induces containment of viral load following ART suspension"

N. DESIDERI, A. BOLASCO, R. FIORAVANTI (2011) "HOMOISOFLAVONOIDS: NATURAL SCAFFOLDS WITH POTENT AND SELECTIVE MONOAMINE OXIDASE-B INHIBITION PROPERTIES"

FABRIZI G, A. GOGGIAMANI (2011) "Heck reaction of arenediazonium salts with N,N-diprotected allylamines. Synthesis of cinnamylamines and indoles."

L. Mannina (2011) "High resolution NMR characterization of olive oils in terms of quality, authenticity and geographical origin"

MAI A, ROTILI D (2011) "Histone deacetylase inhibition modulates deoxyribonucleotide pools and enhances the antitumor effects of the ribonucleotide reductase inhibitor 3'-C-methyladenosine in leukaemia cells."

MATRICARDI P, COVIELLO T (2011) "Hyaluronic acid and Dextran based Semi-IPN Hydrogels as Biomaterials for Bioprinting"

Ragno R, Mai A (2011) "Identification of Small-Molecule Inhibitors of the XendoU Endoribonucleases Family"

Rino Ragno (2011) "Identification of glutathione-methacrylates adducts in gingival fibroblasts and erythrocytes by HPLC-MS and capillary electrophoresis"

Biava (2011) "Identification of potent c-Src inhibitors strongly affecting the proliferation of human neuroblastoma cells"

F. GASPARRINI, P. SIMONE, C. VILLANI, A. CIOGLI (2011) "Immobilized trypsin on epoxy organic monoliths with modulated hydrophilicity: novel bioreactors useful for LC/MS/MS protein analysis"

MATRICARDI P (2011) "In situ forming IPN Hydrogels of calcium alginate and dextran-HEMA for biomedical applications"

G. La Regina, A. Coluccia, R. Silvestri (2011) "Indolylarylsulfones as HIV-1 Non-Nucleoside Reverse Transcriptase Inhibitors: New Cyclic Substituents at the Indole-2-carboxamide."

Baiocco P (2011) "Inhibitory Effect of Silver Nanoparticles on Trypanothione Reductase Activity and Leishmania infantum Proliferation"

MATRICARDI P, DI MEO C, COVIELLO T (2011) "Mechanical characterization of polysaccharide/polyaminoacid hydrogels as potential scaffolds for tissue regeneration"

G. La Regina, R. Silvestri (2011) "Mechanism of interaction of novel indolylarylsulfone derivatives with K103N and Y181I mutant HIV-1 reverse transcriptase in complex with its substrates."

R. Antiochia (2011) "Mediterranean diet and different food models: measurement and comparison of environmental costs using the ecological footprint method"

Mai A, Rotili D (2011) "Modulation of cell differentiation, proliferation, and tumor growth by dihydrobenzyloxopyrimidine non-nucleoside reverse transcriptase inhibitors."

A. MAI (2011) "Modulation of the activity of histone acetyltransferases by long chain alkylidenemalonates (LoCAMs)"

CARLOTTA MARIANECCI, MARIA CARAFA (2011) "Multicompartment vectors as novel drug delivery systems: selective activation of T¿d lymphocytes after zoledronic acid delivery"

Chiara Di Meo (2011) "Mushrooms versus fungi: Natural compounds from Lentinula edodes inhibit aflatoxin biosynthesis by Aspergillus parasiticus"

I. D'ACQUARICA, A. CERRETO, B. BOTTA (2011) "N-Linked peptidoresorc[4]arene-based receptors as noncompetitive inhibitors for a-chymotrypsin"

A. MAI (2011) "N-epsilon-lysine acetylation determines dissociation from GAP junctions and lateralization of connexin 43 in normal and dystrophic heart."

F. Gasparrini, M. Pierini, C. Villani (2011) "NMR and Computational Investigations of the Chiral Discrimination Processes Involving a Cyclic Tetraamidic Chiral Selector"

B. Chiavarino, M. E. Crestoni, S. Fornarini (2011) "Naked Five-Coordinate FeIII(NO) Porphyrin Complexes: Vibrational and Reactivity Features"

A. Ciogli, F. Gasparrini (2011) "New anthranilic acid based antagonists with high affinity and selectivity for the human cholecystokinin receptor 1 (hCCK1-R)"

Valente S, Di Santo R, Costi R, Mai A (2011) "Novel 3,5-bis(bromohydroxybenzylidene)piperidin-4-ones as coactivator-associated arginine methyltransferase 1 inhibitors: enzyme selectivity and cellular activity."

Biava M., Poce G., Alfonso (2011) "Novel Analgesic/Anti-inflammatory Agents: Diarylpyrrole Acetic Esters Endowed with Nitric Oxide Releasing Properties,"

Sergio Valente, Rino Ragno, Antonello Mai (2011) "Novel Cinnamyl Hydroxyamides and 2-Aminoanilides as Histone Deacetylase Inhibitors: Apoptotic Induction and Cytodifferentiation Activity"

CARLOTTA MARIANECCI, FEDERICA RINALDI, M. CARAFA (2011) "Novel pH-sensitive non-ionic surfactant vesicles: comparison between Tween 21 and Tween 20"

Valente S, Mai A. (2011) "Novel reversible monoamine oxidase A inhibitors: highly potent and selective 3-(1H-pyrrol-3-yl)-2-oxazolidinones. "

LA REGINA G., SILVESTRI R. (2011) "Open vessel and cooling while heating microwave-assisted synthesis of pyridinyl N-aryl hydrazones."

A. MAI (2011) "PHARMACOLOGICAL INHIBITION OF HDAC6 ATTENUATES ENDOTHELIAL BARRIER DYSFUNCTION INDUCED BY THROMBIN"

Iazzetti A (2011) "Palladium-Catalyzed Aromatic Sulfonylation: A New Catalytic Domino Process Exploiting in situ Generated Sulfinate Anions "

ROTILI D, MAI A (2011) "Photoactivable peptides for identifying enzyme-substrate and protein-protein interactions."

GABRIELE FAVERO, F. MAZZEI (2011) "Polyazetidine-Coated Microelectrodes: Electrochemical and Diffusion Characterization of Different Redox Substrates"

MATRICARDI P (2011) "Preparation and characterization of a new gellan gum and sulphated hyaluronic acid hydrogel designed for epidural scar prevention"

Luca Pescatori (2011) "Preparation, reactivity and controlled release of SAMs of calix[4,6]arenes and calix[6]arene-based rotaxanes and pseudorotaxanes formed on polycrystalline Cu"

Carlotta Marianecci, Federica Rinaldi, Maria Carafa (2011) "Pulmonary delivery: innovative approaches and perspectives"

Luca Pescatori (2011) "Selective Assembling of Calixarenes and Pseudorotaxanes on Si(100) and Polycrystalline Copper"

ROTILI D., TARANTINO D, MAI A (2011) "Simplification of the tetracyclic SIRT1-selective inhibitor MC2141: coumarin- and pyrimidine-based SIRT1/2 inhibitors with different selectivity profile."

Antonello Mai (2011) "Sirtinol Treatment Reduces Inflammation in Human Dermal Microvascular Endothelial Cells"

Cerreto F., Cesa S., Paolicelli P., Casadei M.A. (2011) "Solid lipid nanoparticles based on low melting lipids as protective system of retinyl palmitate"

I. D'Acquarica, P. Simone, F. Gasparrini, M. Pierini, C Villani (2011) "Stereolability of Dihydroartemisinin, an Antimalarial Drug: A Comprehensive Kinetic Investigation. Part 2"

I. D'ACQUARICA, P. SIMONE, F. GASPARRINI, M. PIERINI, C. VILLANI (2011) "Stereolability of dihydroartemisinin, an antimalarial drug: a comprehensive thermodynamic investigation – Part 1"

Luisa Mannina (2011) "Structural flexibility and role of vicinal 2-thienyl rings in 2,3-dicyano-5,6-di(2-thienyl)-1,4-pyrazine, [(CN)2Th2Pyz], Its palladium(II) complex [(CN)2Th2Pyz(PdCl 2)2], and the related pentametallic pyrazinoporphyrazines [(PdCl2)4Th8TPyzPzM] (M = Mg II(H2O), ZnII)"

Marcello Guidotti (2011) "Sviluppo della definizione di medicinale"

Bruna Bizzarri, Adriana Bolasco, Daniela Secci, Paola Chimenti, Arianna Granese (2011) "Synthesis and biological evaluation of novel 2,4-disubstituted-1,3-thiazoles as anti-Candida spp. agents"

Secci, Carradori, Bolasco, Chimenti (2011) "Synthesis and selective human monoamine oxidase inhibition of 3-carbonyl, 3-acyl, and 3-carboxyhydrazido coumarin derivatives"

ROTILI D, MAI A (2011) "Targeting Histone Demethylases: A New Avenue for the Fight against Cancer."

Luisa Mannina (2011) "Tetra-2,3-pyrazinoporphyrazines with Externally Appended Pyridine Rings. 9. Novel Heterobimetallic Macrocycles and Related Hydrosoluble Hexacations as Potentially Active Photo/Chemotherapeutic Anticancer Agents"

Luisa Mannina (2011) "Tetra-2,3-pyrazinoporphyrazines with externally appended pyridine rings. 11. Photoactivity of a new Pt(II) pentanuclear macrocycle bearing four cisplatin-like functionalities and its related monoplatinated species"

C. FRASCHETTI, M. PIERINI, C. VILLANI, F. GASPARRINI, A. FILIPPI (2011) "The "Bridge" Game: Role of the Fourth Player in Chiral Recognition"

D. Secci, A. Bolasco, P. Chimenti (2011) "The State of the Art of Pyrazole Derivatives as Monoamine Oxidase Inhibitors and Antidepressant/Anticonvulsant Agents"

G. de Petris, A. Cartoni, A. Troiani (2011) "The proton affinity and gas-phase basicity of sulfur dioxide"

F. MAZZEI (2011) "The structure of maize Polyamine Oxidase K300M mutant in complex with the natural substrates provides a snapshot of the catalytic mechanism of polyamine oxidation."

Paolicelli P., Cerreto F., Cesa S., Casadei M.A. (2011) "The system sln-dextran hydrogel: an application for the topical release of ketoconazole"

S. STRANGES (2011) "The valence electronic structure and conformational flexibility of epichlorohydrin"

B. Chiavarino, M. E. Crestoni, S. Fornarini (2011) "Tyrosine nitration as evidenced by IRMPD spectroscopy"

BOTTA B, FRASCHETTI C, D'ACQUARICA I (2011) "Unprecedented gas-phase chiroselective logic gates"

FABRIZI G. (2011) "Update 1 of: Synthesis and Functionalization of Indoles Through Palladium-Catalyzed Reactions"

Franco Mazzei (2011) "Wiring of Redox Enzymes on Three Dimensional Self-Assembled Molecular Scaffold"