IL PORTALE per la RICERCA dei DIPARTIMENTI

Marco Radi (2013) "A Combination Strategy to Inhibit Pim-1: Synergism between Noncompetitive and ATP-Competitive Inhibitors"

A. G. Balducci, F. Sonvico, R. Bettini, P. Colombo, A. Rossi (2013) "Agglomerated Oral Dosage Forms of Artemisinin/ß-cyclodextrin Spray-dried Primary Microparticles Showing Increased Dissolution Rate and Bioavailability "

Marco Radi (2013) "Allosteric Inhibitors of Bcr-Abl: Towards Novel Myristate-Pocket Binders"

Sara Nicoli, Cristina Padula, Patrizia Santi (2013) "Amikacin reverse iontophoresis: Optimization of in vitro extraction"

Incerti M, Tognolini M, Russo S, Pala D, Giorgio C, Hassan-Mohamed I, Vicini P, Piersanti S, Rivara S, Barocelli E, et al. (2013) "Amino acid conjugates of lithocholic acid as antagonists of the EphA2 receptor."

Amori L, Beato C, Costantino G (2013) "Aminonicotinic acid 1-oxides are chemically stable inhibitors of quinolinic acid synthesis in the mammalian brain: a step towards new anti-excitotoxic agents"

Marco Radi (2013) "An alternative synthetic approach for the synthesis of biologically relevant 1,4-disubstituted pyrazolo[3,4-d]pyrimidines"

Mor M (2013) "Antinociceptive effects of the N-acylethanolamine acid amidase inhibitor ARN077 in rodent pain models"

Dell'Amico Luca (2013) "Asymmetric Organocatalytic Benzylation of a,ß-Unsaturated Aldehydes with Toluenes"

Dell'Amico Luca (2013) "Beyond classical reactivity patterns: shifting from 1,4- to 1,6-additions in regio- and enantioselective organocatalyzed vinylogous reactions of olefinic lactones with enals and 2,4-dienals"

S. Bruno, A. Mozzarelli (2013) "CO rebinding kinetics and molecular dynamics simulations highlight dynamic regulation of internal cavities in human cytoglobin"

Lodola A (2013) "Conformational effects on the pro-S hydrogen abstraction reaction in cyclooxygenase-1: an integrated QM/MM and MD study."

Marco Radi (2013) "Design, Synthesis, and Biological Evaluation of Pyrazolo[3,4-d]pyrimidines Active in Vivo on the Bcr-Abl T315I Mutant"

Cristina Padula, Patrizia Santi (2013) "Development of a Doxazosin and Finasteride Transdermal System for Combination Therapy of Benign Prostatic Hyperplasia"

M. Tognolini (2013) "Dietary (Poly)phenolics in Human Health: Structures, Bioavailability and Evidence of Protective Effects Against Chronic Diseases"

Elda Favari, Francesca Zimetti, Franco Bernini (2013) "Differential effects of fenofibrate and extended-release niacin on high-density lipoprotein particle size distribution and cholesterol efflux capacity in dyslipidemic patients"

Mor M (2013) "Discovery of a New Class of Highly Potent Inhibitors of Acid Ceramidase: Synthesis and Structure-Activity Relationship (SAR)."

S. PESCINA, S. NICOLI (2013) "Drug adsorption on bovine and porcine sclera studied with streaming potential"

C. Padula, P. Santi, F. Sonvico, S. Barbieri (2013) "Dynamics of water and small molecules in bioadhesive polymer films"

Silvia Pescina, Patrizia Santi, Sara Nicoli (2013) "Effect of iontophoresis on the in vitro trans-scleral transport of three single stranded oligonucleotides"

F. BUTTINI, P. COLOMBO (2013) "Effect of polymers for aerolization properties of mannitol-based microcomposites containing meloxicam"

M. Mor (2013) "Epidermal growth factor receptor tyrosine kinase inhibitors: current status and future perspectives in the development of novel irreversible inhibitors for the treatment of mutant non-small cell lung cancer"

A. Mozzarelli, B. Campanini (2013) "Fine tuning of the active site modulates specificity in the interaction of O-acetylserine sulfhydrylase isozymes with serine acetyltransferase"

G. Costantino, M. Mor (2013) "Further insights in 5-phenyl-2-[2-(1-piperidinylcarbonyl) phenyl]-2,3-dihydro-1H-pyrrolo[1,2-c]imidazol-1-ones, a recently disclosed class of Neuropeptide S antagonists"

Colombo P (2013) "Group A2 Analogs of Innovator Teicoplanin: Variability of their Ratio during Treatment Time Course in Human Blood; Consequences for the Generics"

Cristina Padula, Sara Nicoli, Patrizia Santi (2013) "In Vitro Evaluation of Mucoadhesive Films for Gingival Administration of Lidocaine"

S. PESCINA, P. SANTI, C. PADULA, S. NICOLI (2013) "In vitro trans-scleral iontophoresis of methylprednisolone hemisuccinate with short application time and high drug concentration"

R. Bettini, F. Sonvico, P. Colombo (2013) "Investigation of the swelling behavior of Dome Matrix drug delivery modules by high-resolution X-ray computed tomography"

Campanini B, Raboni S, Mozzarelli A. (2013) "Isozyme-specific ligands for O-acetylserine sulfhydrylase, a novel antibiotic target"

C. Padula, P. Santi (2013) "Liposomal-benzocaine gel formulation: correlation between in vitro assays and in vivo topical anesthesia in volunteers"

C. Carmi, M. Mor (2013) "Molecular mechanisms underlying the antitumor activity of 3-aminopropanamide irreversible inhibitors of the epidermal growth factor receptor in non-small cell lung cancer"

Paolo Colombo (2013) "Multiple dosing of simvastatin inhibits airway mucus production of epithelial cells: Implications in the treatment of chronic obstructive airway pathologies"

Paredi GL, Mozzarelli A (2013) "Muscle and meat: New horizons and applications for proteomics on a farm to fork perspective"

F. Sonvico (2013) "Nanomedical research in Australia and New Zealand"

Lodola Alessio, Mor Marco (2013) "Nonempirical energetic analysis of reactivity and covalent inhibition of fatty acid amide hydrolase."

Barocelli E (2013) "Polyunsaturated fatty acid metabolism signature in ischemia differs from reperfusion in mouse intestine.."

Marco Radi (2013) "Pyrazolo[3,4-d]pyrimidine Prodrugs: Strategic Optimization of the Aqueous Solubility of Dual Src/Abl Inhibitors"

Lodola A, Rivara S, Mor M. (2013) "Quantum mechanics/molecular mechanics modeling of fatty acid amide hydrolase reactivation distinguishes substrate from irreversible covalent inhibitors."

Costantino G (2013) "State of-the-art and dissemination of computational tools for drug-design purposes: a survey among Italian academics and industrial institutions."

Cristina Padula, Patrizia Santi (2013) "Strategies for delivering local anesthetics to the skin: focus on liposomes, solid lipid nanoparticles, hydrogels and patches"

Pala D, Lodola A, Rivara S, Mor M. (2013) "Structure-based virtual screening of MT2 melatonin receptor: influence of template choice and structural refinement."

Marco Mor (2013) "Synthesis and Structure–Activity Relationship (SAR) of 2-Methyl-4-oxo-3-oxetanylcarbamic Acid Esters, a Class of PotentN-Acylethanolamine Acid Amidase (NAAA) Inhibitors"

Marco Mor (2013) "Synthesis and Structure–Activity Relationship Studies ofO-Biphenyl-3-yl Carbamates as Peripherally Restricted Fatty Acid Amide Hydrolase Inhibitors"

A. Mozzarelli (2013) "Tertiary and quaternary allostery in tetrameric hemoglobin from Scapharca inaequivalvis"

Colombo P (2013) "Towards the Bioequivalence of Pressurised Metered Dose Inhalers 2. Aerodynamically equivalent particles (with and without glycerol) exhibit different biopharmaceutical profiles in vitro"

Costantino G (2013) "Unbinding pathways from the glucocorticoid receptor shed light on the reduced sensitivity of glucocorticoid ligands to a naturally occurring, clinically relevant mutant receptor"

Marco Radi (2013) "Unconventional plasticity of hiv-1 reverse transcriptase: How inhibitors could open a connection "gate" between allosteric and catalytic sites"

Mozzarelli A (2013) "Unintended consequences? Water molecules at biological and crystallographic protein–protein interfaces"